SCHEMBL12470609

SCHEMBL12470609

CC(C)(C)OC(=O)Nc1ccc2c(c1)C(=O)CC(C)(C)S2(=O)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 2/20 0.41
CA1 P00915 2/20 0.41
CA9 Q16790 2/20 0.41
SLC10A2 Q12908 1/20 0.40
BRD4 O60885 2/20 0.38
CREBBP Q92793 2/20 0.38
PSMB8 P28062 1/20 0.37
HCRTR1 O43613 1/20 0.36
HCRTR2 O43614 1/20 0.36
PRKDC P78527 1/20 0.36
CA2 P00918 1/20 0.36
SIRT2 Q8IXJ6 1/20 0.36
SIRT1 Q96EB6 1/20 0.36
BUB1 O43683 1/20 0.36
CYP17A1 P05093 1/20 0.36
IDH1 O75874 1/20 0.35
ALDH1A1 P00352 1/20 0.35
GAA P10253 1/20 0.35
ABCC9 O60706 1/20 0.35
ABCC8 Q09428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11904283 0.79 CA12 (0.43) CA12CA1CA9SLC10A2BRD4
SCHEMBL29921889 0.76 CA12 (0.47) CA12CA1CA9BRD4CREBBP
SCHEMBL12470984 0.75 CA12 (0.42) CA12CA1CA9BRD4CREBBP
SCHEMBL11904033 0.75 MAPT (0.53) CA12CA1CA9SIRT2SIRT1
SCHEMBL29921932 0.73 KDM4E (0.53) CA12CA1CA9SIRT2SIRT1
SCHEMBL15022432 0.72 MAPT (0.52) CA12CA1CA9BRD4CREBBP
SCHEMBL7235169 0.69 BAZ2B (0.52) CA12CA1CA9ACHEBACE1
SCHEMBL20809725 0.69 BAZ2B (0.55) CA12CA1CA9NR1I3
SCHEMBL30781540 0.69 BAZ2B (0.55) CA12CA1CA9NR1I3
SCHEMBL4314672 0.69 CA12 (0.49) CA12CA1CA9PSMB8PRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012107262-A1 DIHYDROBENZOPYRAN, THIOCHROMAN, TETRAHYDROQUINOLEINE AND TETRAHYDRONAPHTALENE DERIVATIVES AND THEIR USE IN ANTICANCER THERAPY UNIVERSITE DE LIEGE (BE) 2012-08-16 WO disclosed