SCHEMBL12475441

SCHEMBL12475441

O=S(=O)(O)CCc1ccc2c(c1)B(O)OC2

nearest known ligand 0.56

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA12 O43570 10/20 0.49
CA1 P00915 10/20 0.49
CA2 P00918 10/20 0.49
CA9 Q16790 10/20 0.49
CA4 P22748 7/20 0.49
KLK1 P06870 1/20 0.44
KLK5 Q9Y337 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15981493 0.79 CA1 (0.63) CA12CA1CA2CA9CA4
SCHEMBL12383669 0.78 CA1 (0.55) CA12CA1CA2CA9CA4
SCHEMBL22847886 0.75 CA1 (0.57) CA12CA1CA2CA9CA4
SCHEMBL12475507 0.75 ROCK2 (0.64) CA12CA1CA2CA9CA4
SCHEMBL18500989 0.75 CA1 (0.53) CA12CA1CA2CA9CA4
SCHEMBL2299412 0.75 CA12 (0.60) CA12CA1CA2CA9CA4
SCHEMBL14986243 0.72 CA1 (0.53) CA12CA1CA2CA9CA4
SCHEMBL12383659 0.72 KLK5 (0.56) CA12CA1CA2CA9CA4
SCHEMBL12383358 0.72 CA1 (0.53) CA12CA1CA2CA9CA4
SCHEMBL20607758 0.71 CA1 (0.60) CA12CA1CA2CA9CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2673281-A1 BORON CONTAINING POLYBASIC BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTICS USES THEREOF Rempex Pharmaceuticals, Inc. (US) 2013-12-18 EP disclosed
WO-2012109164-A1 BORON CONTAINING POLYBASIC BACTERIAL EFFLUX PUMP INHIBITORS AND THERAPEUTICS USES THEREOF REMPEX PHARMACEUTICALS, INC. (US) 2012-08-16 WO disclosed