SCHEMBL1247558

SCHEMBL1247558

Cc1onc(-c2ccc(Oc3cccc(CC(=O)O)c3)cc2)c1NC(=O)OCCc1ccccc1F

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 6/20 0.42
SCN5A Q14524 4/20 0.42
NPSR1 Q6W5P4 1/20 0.41
MAPT P10636 1/20 0.40
PPARG P37231 2/20 0.40
PPARD Q03181 2/20 0.40
PPARA Q07869 2/20 0.40
NTRK1 P04629 2/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.38
PTGDR2 Q9Y5Y4 1/20 0.38
TDP1 Q9NUW8 1/20 0.37
FFAR1 O14842 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1247800 0.93 SCN9A (0.42) SCN9ASCN5ANPSR1MAPTNTRK1
SCHEMBL1245138 0.92 SCN9A (0.52) SCN9ASCN5ANPSR1MAPTPPARG
SCHEMBL1245272 0.88 SCN9A (0.45) SCN9ASCN5ANPSR1MAPTPPARG
SCHEMBL3712293 0.87 LPAR1 (0.49) MAPTPPARGPPARDPPARANPC1
SCHEMBL1246481 0.84 SCN9A (0.54) SCN9ASCN5ANPSR1MAPTPPARD
SCHEMBL11896062 0.83 LPAR1 (0.47) SCN9ASCN5ANPSR1MAPTALDH1A1
SCHEMBL1247570 0.83 SCN9A (0.46) SCN9ASCN5ANPSR1MAPTNTRK1
SCHEMBL1246308 0.82 SCN9A (0.55) SCN9ASCN5ANPSR1NTRK1TDP1
SCHEMBL1246915 0.82 SCN9A (0.41) SCN9ASCN5ANPSR1MAPTPPARG
SCHEMBL9902692 0.82 SCN9A (0.40) SCN9ASCN5ANPSR1MAPTNTRK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2462128-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS Amira Pharmaceuticals, Inc. (US) 2012-06-13 EP claimed
WO-2011017350-A2 COMPOUNDS AS LYSOPHOSPHATIDIC ACID RECEPTOR ANTAGONISTS AMIRA PHARMACEUTICALS, INC. (US) 2011-02-10 WO claimed