SCHEMBL12487404

SCHEMBL12487404

CCc1nc(N)nc(N)c1OCCCOc1cccc(-c2c(N)nc(N)nc2CC)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHFR P00374 16/20 1.00
HEXA P06865 2/20 0.58
HEXB P07686 2/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12487396 0.85 DHFR (1.00) DHFRHEXAHEXB
Hydrochloric Acid SCHEMBL12486624 0.84 DHFR (1.00) DHFRHEXAHEXB
SCHEMBL31155861 0.80 DHFR (0.70) DHFR
SCHEMBL12487635 0.79 DHFR (1.00) DHFRHEXAHEXB
SCHEMBL31155805 0.77 DHFR (0.62) DHFR
SCHEMBL31155835 0.76 DHFR (0.66) DHFR
Hydrochloric Acid SCHEMBL31155866 0.76 DHFR (0.64) DHFR
SCHEMBL31155847 0.76 DHFR (0.63) DHFR
SCHEMBL12368253 0.74 HEXA (1.00) DHFRHEXAHEXB
SCHEMBL31155783 0.74 DHFR (0.58) DHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012121682-A2 ANTI-FOLATE ANTIMALARIALS WITH DUAL-BINDING MODES AND THEIR PREPARATION NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2012-09-13 WO claimed
US-9000003-B2 Anti-folate antimalarials with dual-binding modes and their preparation NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2015-04-07 US disclosed
US-9000003-B2 Anti-folate antimalarials with dual-binding modes and their preparation NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2015-04-07 US disclosed
WO-2012121682-A2 ANTI-FOLATE ANTIMALARIALS WITH DUAL-BINDING MODES AND THEIR PREPARATION NATIONAL SCIENCE AND TECHNOLOGY DEVELOPMENT AGENCY (TH) 2012-09-13 WO disclosed