SCHEMBL12489602

SCHEMBL12489602

Nc1nccc(-n2ncc3ccccc32)n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 6/20 0.56
CDK2 P24941 6/20 0.56
ROCK1 Q13464 3/20 0.56
CCNT1 O60563 2/20 0.52
CDK1 P06493 2/20 0.52
CCNB1 P14635 2/20 0.52
CDK9 P50750 2/20 0.52
CDK7 P50613 1/20 0.52
CCNH P51946 1/20 0.52
PAK4 O96013 1/20 0.52
PIKFYVE Q9Y2I7 1/20 0.52
MKNK1 Q9BUB5 1/20 0.51
MKNK2 Q9HBH9 1/20 0.51
MAPK8 P45983 1/20 0.51
MAPK9 P45984 1/20 0.51
MAPK10 P53779 1/20 0.51
TTBK1 Q5TCY1 4/20 0.49
TTBK2 Q6IQ55 1/20 0.46
MAP3K14 Q99558 1/20 0.46
LRRK2 Q5S007 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12525017 0.81 PAK4 (0.59) CDC7CDK2PAK4PIKFYVETTBK1
SCHEMBL30459875 0.81 MKNK1 (0.51) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL17683140 0.81 MKNK1 (0.51) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL11970748 0.79 PAK4 (0.57) CDC7CDK2ROCK1PAK4PIKFYVE
SCHEMBL11970491 0.79 MAP3K14 (0.60) CDC7CDK2ROCK1PAK4PIKFYVE
SCHEMBL3824181 0.77 MKNK1 (0.48) CDC7CDK2ROCK1CCNT1CDK1
SCHEMBL12075159 0.77 MKNK1 (0.46) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL31020506 0.76 IRAK4 (0.57) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL12075537 0.76 IRAK4 (0.57) CCNT1CDK1CCNB1CDK9CDK7
SCHEMBL11970828 0.76 PAK4 (0.66) CDC7CDK2PAK4PIKFYVETTBK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2686314-A1 6,5-HETEROCYCLIC PROPARGYLIC ALCOHOL COMPOUNDS AND USES THEREFOR F.HOFFMANN-LA ROCHE AG (CH) 2014-01-22 EP disclosed
WO-2012123522-A1 6,5-HETEROCYCLIC PROPARGYLIC ALCOHOL COMPOUNDS AND USES THEREFOR F. HOFFMANN-LA ROCHE AG (CH) 2012-09-20 WO disclosed