SCHEMBL12489705

SCHEMBL12489705

COc1cccc2c[n+](O)ccc12

nearest known ligand 0.50

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ACHE P22303 18/20 0.50
BCHE P06276 13/20 0.50
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
HPGD P15428 1/20 0.45
HSD17B10 Q99714 1/20 0.45
NQO1 P15559 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11960608 0.86 ACHE (0.62) ACHEBCHE
SCHEMBL10262042 0.80 ACHE (0.47) ACHEBCHENQO1
SCHEMBL754022 0.79 ACHE (0.46) ACHEBCHENQO1
SCHEMBL18526636 0.79 ACHE (0.48) ACHEBCHENQO1
SCHEMBL12844094 0.78 MAPT (0.46) ACHEBCHEKDM4EALDH1A1HPGD
SCHEMBL8244435 0.76 CYP19A1 (0.40) ACHEBCHEKDM4EHPGD
SCHEMBL13219676 0.76 CYP2A6 (0.50) ACHEALDH1A1HPGDHSD17B10
SCHEMBL29367279 0.72 MAPT (0.61) ACHEBCHEKDM4EALDH1A1HSD17B10
SCHEMBL30373629 0.72 MAPT (0.61) ACHEBCHEKDM4EALDH1A1HSD17B10
SCHEMBL151449 0.72 MAPT (0.61) ACHEBCHEKDM4EALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2328865-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2017-05-31 EP disclosed
EP-2414350-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2014-11-12 EP disclosed
EP-2414352-B1 HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2014-10-01 EP disclosed
WO-2011082077-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-07-07 WO disclosed
WO-2011075439-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-06-23 WO disclosed
WO-2011059887-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed
WO-2011059850-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed
WO-2010138368-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-12-02 WO disclosed
WO-2010138488-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2010-12-02 WO disclosed