SCHEMBL12499752

SCHEMBL12499752

O=C(O)c1c(C2CCC2)cnc2[nH]ncc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 2/20 0.43
CCNE1 P24864 3/20 0.40
CDK2 P24941 3/20 0.40
CCNE2 O96020 2/20 0.40
CCNB2 O95067 1/20 0.40
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
CCNB3 Q8WWL7 1/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
HPGDS O60760 1/20 0.38
HCAR2 Q8TDS4 1/20 0.37
TRPV1 Q8NER1 4/20 0.35
SGK1 O00141 1/20 0.35
AURKA O14965 1/20 0.35
CAMKK1 Q8N5S9 1/20 0.35
SGK3 Q96BR1 1/20 0.35
CAMKK2 Q96RR4 1/20 0.35
SGK2 Q9HBY8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1695107 0.85 HTR1D (0.42) JAK3CCNE1CDK2CCNE2CCNB2
SCHEMBL3730728 0.69 AKT2 (0.39) JAK3JAK2JAK1TYK2HPGDS
Hydrochloric Acid SCHEMBL3716590 0.68 AKT2 (0.39) JAK3JAK2JAK1TYK2HPGDS
SCHEMBL3739352 0.68 JAK1 (0.44) JAK3JAK2JAK1TYK2TSHR
SCHEMBL4340262 0.67 PDE4B (0.54) JAK3CCNE1CDK2CCNE2CCNB2
SCHEMBL15007485 0.66 RPS6KA3 (0.44) JAK3CCNE1CDK2CCNE2CCNB2
SCHEMBL285566 0.66 CCNE2 (0.42) CCNE1CDK2CCNE2CCNB2CDK1
SCHEMBL17105468 0.65 HCAR2 (0.35) HCAR2CAMKK2SMN1; SMN2
SCHEMBL21157774 0.64 CDK2 (0.46) JAK3CCNE1CDK2CCNE2CCNB2
SCHEMBL22018238 0.64 CDK2 (0.46) JAK3CCNE1CDK2CCNE2CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2681216-A2 SUBSTITUTED 6,5-FUSED BICYCLIC HETEROARYL COMPOUNDS Epizyme, Inc. (US) 2014-01-08 EP disclosed
WO-2012118812-A2 SUBSTITUTED 6,5-FUSED BICYCLIC HETEROARYL COMPOUNDS Epizyme, Inc. (US) 2012-09-07 WO disclosed