SCHEMBL12499754

SCHEMBL12499754

N/C(Cc1ccc(Cl)c(Cl)c1)=C(\C(=O)O)C(=O)C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.40
LMNA P02545 3/20 0.40
HSP90AA1 P07900 2/20 0.40
PIK3CA P42336 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.39
CA2 P00918 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
BLM P54132 1/20 0.38
POLB P06746 1/20 0.38
HAO1 Q9UJM8 1/20 0.38
CCR2 P41597 4/20 0.38
IDO1 P14902 1/20 0.37
GAA P10253 1/20 0.37
CRHBP P24387 1/20 0.37
CRHR2 Q13324 1/20 0.37
PDPK1 O15530 1/20 0.36
S1PR5 Q9H228 1/20 0.36
MEN1 O00255 1/20 0.36
MAPT P10636 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12499758 1.00 KMT2A (0.40) KMT2ALMNAHSP90AA1PIK3CALOXL2
SCHEMBL12499895 0.84 CTBP2 (0.44) KMT2ALMNAALDH1A1POLBMEN1
SCHEMBL12498657 0.84 CTBP2 (0.44) KMT2ALMNAALDH1A1POLBMEN1
SCHEMBL12498763 0.82 CTBP2 (0.50) KMT2APIK3CAKDM4EALDH1A1MEN1
SCHEMBL12498765 0.82 CTBP2 (0.50) KMT2APIK3CAKDM4EALDH1A1MEN1
SCHEMBL12498668 0.78 PIK3CA (0.42) PIK3CAIDO1PDPK1
SCHEMBL12498667 0.78 PIK3CA (0.42) PIK3CAIDO1PDPK1
Trifluoroacetic Acid SCHEMBL3399696 0.78 SLC6A4 (0.46) KMT2ALMNAHSP90AA1PIK3CACA2
SCHEMBL12499833 0.77 MEN1 (0.51) KMT2AALDH1A1IDO1MEN1MAPT
SCHEMBL12499832 0.77 MEN1 (0.51) KMT2AALDH1A1IDO1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012103071-A2 COMPOUNDS AND COMPOSITIONS EISAI R&D MANAGEMENT CO., LTD. (JP) 2012-08-02 WO disclosed