SCHEMBL12501693

SCHEMBL12501693

CC(C)(C)OC(=O)N1CCC[C@@H](C(=O)Nc2cc(-c3cc(F)ncc3Cl)c(Cl)cn2)C1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CDK9 P50750 15/20 0.51
CDK1 P06493 2/20 0.45
CDK4 P11802 2/20 0.45
CDK2 P24941 2/20 0.45
CCNT1 O60563 7/20 0.44
NTRK1 P04629 1/20 0.44
MAPK8 P45983 3/20 0.43
MAPK10 P53779 3/20 0.43
MAPK14 Q16539 3/20 0.43
CCNB1 P14635 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK7 P50613 1/20 0.43
CCNH P51946 1/20 0.43
MNAT1 P51948 1/20 0.43
CDK3 Q00526 1/20 0.43
CDK6 Q00534 1/20 0.43
CDK5 Q00535 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12501692 1.00 CDK9 (0.51) CDK9CDK1CDK4CDK2CCNT1
SCHEMBL1944753 0.87 CCNT1 (0.54) CDK9CDK4CDK2CCNT1NTRK1
SCHEMBL1944749 0.87 CCNT1 (0.54) CDK9CDK4CDK2CCNT1NTRK1
SCHEMBL1439644 0.87 CDK9 (0.55) CDK9CDK1CDK4CDK2CCNT1
SCHEMBL1439640 0.87 CDK9 (0.55) CDK9CDK1CDK4CDK2CCNT1
SCHEMBL1439849 0.86 USP30 (0.50) CDK9CCNT1MAPK8MAPK10MAPK14
SCHEMBL1439848 0.86 USP30 (0.50) CDK9CCNT1MAPK8MAPK10MAPK14
SCHEMBL12827050 0.86 CDK9 (0.46) CDK9NTRK1MAPK8MAPK10MAPK14
SCHEMBL16042236 0.85 CDK9 (0.46) CDK9NTRK1MAPK8MAPK10MAPK14
SCHEMBL16042238 0.85 CDK9 (0.46) CDK9NTRK1MAPK8MAPK10MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101063-A1 N-ACYL PYRIDINE BIARYL COMPOUNDS AND THEIR USES NOVARTIS AG (CH) 2012-08-02 WO disclosed