SCHEMBL12520141

SCHEMBL12520141

c1cncc(OC2CCCCC2)c1

nearest known ligand 0.67

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 3/20 0.67
CHRNA4 P43681 3/20 0.67
CYP11B2 P19099 1/20 0.50
MKNK1 Q9BUB5 1/20 0.47
MKNK2 Q9HBH9 1/20 0.47
ALDH1A1 P00352 2/20 0.46
HTT P42858 1/20 0.46
CHRNA3 P32297 2/20 0.45
CHRNA7 P36544 2/20 0.45
CHRNA1 P02708 1/20 0.45
CHRNG P07510 1/20 0.45
CHRNB1 P11230 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRND Q07001 1/20 0.45
GRM2 Q14416 1/20 0.45
EPHX2 P34913 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2083914 0.98 CHRNB2 (0.69) CHRNB2CHRNA4CYP11B2MKNK1MKNK2
SCHEMBL12949446 0.94 CHRNB2 (0.69) CHRNB2CHRNA4MKNK1MKNK2CHRNA3
Hydrochloric Acid SCHEMBL29877020 0.93 CHRNB2 (0.67) CHRNB2CHRNA4MKNK1MKNK2CHRNA3
Hydrochloric Acid SCHEMBL16823577 0.93 CHRNB2 (0.67) CHRNB2CHRNA4MKNK1MKNK2CHRNA3
SCHEMBL31276985 0.90 CHRNB2 (0.67) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL16845110 0.90 CHRNB2 (0.67) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
Hydrochloric Acid SCHEMBL16823600 0.89 CHRNB2 (0.65) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1
SCHEMBL3825648 0.85 CHRNB2 (0.70) CHRNB2CHRNA4MKNK1MKNK2CHRNA3
SCHEMBL7788072 0.84 CHRNB2 (0.78) CHRNB2CHRNA4MKNK1MKNK2CHRNA3
SCHEMBL3122156 0.84 CHRNB2 (0.59) CHRNB2CHRNA4CHRNA3CHRNA7CHRNA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2523951-B1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES INC (US) 2015-04-22 EP disclosed
WO-2011088303-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES , INC. (US) 2011-07-21 WO disclosed
WO-2011011303-A1 INHIBITORS OF FLAVIVIRIDAE VIRUSES GILEAD SCIENCES, INC. (US) 2011-01-27 WO disclosed