SCHEMBL12526432

SCHEMBL12526432

O=C(CNCO)Nc1cccc(C(F)(F)F)c1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.67
MEN1 O00255 5/20 0.67
KMT2A Q03164 5/20 0.67
GAA P10253 2/20 0.67
XBP1 P17861 1/20 0.67
NPSR1 Q6W5P4 1/20 0.67
L3MBTL1 Q9Y468 2/20 0.65
HTT P42858 2/20 0.65
SMN1; SMN2 Q16637 1/20 0.63
ALDH1A1 P00352 3/20 0.62
HDAC3 O15379 1/20 0.60
HDAC1 Q13547 1/20 0.60
HDAC2 Q92769 1/20 0.60
HDAC10 Q969S8 1/20 0.60
HDAC11 Q96DB2 1/20 0.60
HDAC8 Q9BY41 1/20 0.60
HDAC6 Q9UBN7 1/20 0.60
NCOR2 Q9Y618 1/20 0.60
RAB9A P51151 1/20 0.59
LMNA P02545 2/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12020641 0.86 MAPT (0.60) MAPTMEN1KMT2AGAAXBP1
SCHEMBL693942 0.86 MAPT (0.72) MAPTMEN1KMT2AGAAXBP1
SCHEMBL5142590 0.85 MAPT (0.77) MAPTMEN1KMT2AGAAXBP1
SCHEMBL31236338 0.85 MAPT (0.77) MAPTMEN1KMT2AGAAXBP1
SCHEMBL966420 0.85 SMN1; SMN2 (0.68) MAPTMEN1KMT2AGAAXBP1
SCHEMBL5355449 0.84 L3MBTL1 (0.64) MAPTMEN1KMT2AGAAXBP1
SCHEMBL21580306 0.84 HTT (0.76) MAPTMEN1KMT2AGAAXBP1
SCHEMBL963689 0.83 HDAC3 (0.70) MAPTMEN1KMT2AGAAXBP1
SCHEMBL26627751 0.83 MAPT (0.72) MAPTMEN1KMT2AGAAXBP1
SCHEMBL693941 0.83 MAPT (0.72) MAPTMEN1KMT2AGAAXBP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012125661-A1 SUBSTITUTED 3-AZABICYCLO[3.1.0]HEXANE DERIVATIVES USEFUL AS CCR2 ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2012-09-20 WO disclosed