SCHEMBL12528516

SCHEMBL12528516

C=CCCN(Cc1ccccc1)C(=O)[C@H](CC=C)NC(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
USP2 O75604 2/20 0.45
AKT1 P31749 2/20 0.45
CTSS P25774 5/20 0.44
CTSK P43235 3/20 0.44
CTSL P07711 2/20 0.44
CTSB P07858 2/20 0.44
PPARA Q07869 2/20 0.43
PPARG P37231 1/20 0.43
ACE P12821 1/20 0.43
PSEN1 P49768 2/20 0.42
PSEN2 P49810 2/20 0.42
APH1B Q8WW43 2/20 0.42
NCSTN Q92542 2/20 0.42
APH1A Q96BI3 2/20 0.42
PSENEN Q9NZ42 2/20 0.42
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18342602 0.82 ACE (0.46) AKT1CTSSCTSKCTSLCTSB
SCHEMBL1341914 0.79 PPARA (0.57) USP2CTSSPPARAPPARG
SCHEMBL1343633 0.79 PPARA (0.57) USP2CTSSPPARAPPARG
SCHEMBL14085940 0.79 CTSS (0.52) AKT1CTSSCTSKCTSLCTSB
SCHEMBL1007073 0.78 CTSS (0.49) USP2AKT1CTSSCTSKCTSL
SCHEMBL1007074 0.78 CTSS (0.49) USP2AKT1CTSSCTSKCTSL
SCHEMBL3107411 0.77 PPARA (0.51) CTSSCTSKCTSLCTSBPPARA
SCHEMBL18526468 0.77 PPARA (0.55) CTSSCTSKCTSLCTSBPPARA
SCHEMBL15071347 0.77 CTSS (0.50) AKT1CTSSCTSKCTSLCTSB
SCHEMBL12527921 0.76 CTSS (0.45) CTSSCTSKCTSLCTSBPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9346852-B2 Substituted adipic acid amides and uses thereof BRISTOL-MYERS SCUIBB COMPANY (US) 2016-05-24 US disclosed
US-9346852-B2 Substituted adipic acid amides and uses thereof BRISTOL-MYERS SCUIBB COMPANY (US) 2016-05-24 US disclosed
WO-2012125622-A1 SUBSTITUTED ADIPIC ACID AMIDES AND USES THEREOF BRISTOL-MYERS SQUIBB COMPANY (US) 2012-09-20 WO disclosed