SCHEMBL125495

SCHEMBL125495

Nc1ccc(N)c2c1C(=O)c1c(N)ccc(N)c1C2=O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 3/20 1.00
CSNK2A2 P19784 1/20 0.70
CSNK2B P67870 1/20 0.70
CSNK2A1 P68400 1/20 0.70
CSNK2A3 Q8NEV1 1/20 0.70
ADORA2A P29274 4/20 0.65
CSNK1A1 P48729 2/20 0.65
CSNK1D P48730 2/20 0.65
CSNK1G1 Q9HCP0 2/20 0.65
MAOA P21397 2/20 0.65
FGR P09769 1/20 0.65
PIM1 P11309 1/20 0.65
DYRK1A Q13627 1/20 0.65
HIPK2 Q9H2X6 1/20 0.65
MEN1 O00255 6/20 0.50
KMT2A Q03164 6/20 0.50
POLB P06746 4/20 0.50
ALDH1A1 P00352 3/20 0.50
MAPT P10636 3/20 0.50
TDP1 Q9NUW8 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29378892 1.00 THRB (1.00) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL29390741 1.00 THRB (1.00) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL14750382 0.86 THRB (0.74) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL8577844 0.86 THRB (0.74) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL3843709 0.84 CSNK2A2 (1.00) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL10355835 0.84 ADORA2A (0.73) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL9619698 0.84 THRB (0.70) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL10356104 0.84 ADORA2A (0.73) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL498572 0.84 CSNK2A2 (1.00) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3
SCHEMBL504614 0.84 CSNK2A2 (1.00) THRBCSNK2A2CSNK2BCSNK2A1CSNK2A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 2259 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025149345-A1 LAUNDRY DETERGENT PRODUCT UNILEVER IP HOLDINGS B.V. (NL) 2025-07-17 WO claimed
WO-2025109628-A1 A SYNERGISTIC TERNARY INSECTICIDAL COMPOSITION RAJDHANI PETROCHEMICALS PRIVATE LIMITED (IN) 2025-05-30 WO claimed
US-20250075051-A1 PROCESS FOR RECYCLING CONTAMINATED POLYMERS ARKEMA FRANCE (FR) 2025-03-06 US claimed
CN-114981395-B Laundry detergent product 联合利华知识产权控股有限公司 2024-11-26 CN claimed
EP-4457275-A1 PROCESS FOR RECYCLING CONTAMINATED POLYMERS ARKEMA FRANCE (FR) 2024-11-06 EP claimed
US-12130267-B2 Analyzing method for azo compound SHIMADZU CORPORATION (JP) 2024-10-29 US claimed
WO-2024100569-A1 SUNSCREEN FORMULATION COMPRISING MICROCAPSULES, AND PROCESS FOR MANUFACTURING SUCH MICROCAPSULES COSMETIC DEVELOPMENT GROUP (FR) 2024-05-16 WO claimed
CN-117820586-A Cationic waterborne polyurethane type macromolecular dye and preparation method thereof 香港理工大学深圳研究院 2024-04-05 CN claimed
US-20230407208-A1 LAUNDRY DETERGENT PRODUCT CONOPCO, INC., D/B/A UNILEVER (US) 2023-12-21 US claimed
US-20230292753-A1 AN INSECTICIDAL COMPOSITION FOR PEST CONTROL COMPRISING OF DIACYLHYDRAZINES RAJDHANI PETROCHEMICALS PRIVATE LIMITED (IN) 2023-09-21 US claimed
EP-0012965-B1 PRODUCT AND PROCESS FOR DYEING HAIR Wella Aktiengesellschaft (DE) 1982-08-25 EP claimed
EP-0043436-A1 Composition and process for dyeing hair Wella Aktiengesellschaft (DE) 1982-01-13 EP claimed
US-4279613-A 4-ISOPROPYL CRESOL COUPLER AND DEVELOPER THEREFOR WELLA AKTIENGESELLSCHAFT (DE) 1981-07-21 US claimed
EP-0008080-B1 HAIR DYEING COMPOSITION Wella Aktiengesellschaft (DE) 1981-07-01 EP claimed
EP-0012965-A1 Product and process for dyeing hair Wella Aktiengesellschaft (DE) 1980-07-09 EP claimed
WO-1980001241-A1 COMPOSITION AND PROCESS FOR HAIR COLOURATION WELLA AG (DE) 1980-06-26 WO claimed
WO-1980000417-A1 PREPARATION FOR HAIR COLORATION WELLA AG (DE) 1980-03-20 WO claimed
WO-1980000303-A1 PREPARATION FOR HAIR COLORATION WELLA AG (DE) 1980-03-06 WO claimed
EP-0008080-A2 Hair dyeing composition Wella Aktiengesellschaft (DE) 1980-02-20 EP claimed
EP-0008039-A1 Hair dyeing composition containing 6-amino-3-methyl-phenol Wella Aktiengesellschaft (DE) 1980-02-20 EP claimed