SCHEMBL12558658

SCHEMBL12558658

Oc1ccc(C2C(O)CN(P)CC2O)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 13/20 0.39
ESR1 P03372 6/20 0.33
CYP2C9 P11712 2/20 0.33
KDM1A O60341 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP3A4 P08684 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.32
CA12 O43570 1/20 0.32
GMNN O75496 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
LMNA P02545 1/20 0.32
CA3 P07451 1/20 0.32
MAPT P10636 1/20 0.32
TYR P14679 1/20 0.32
HPGD P15428 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12558167 0.85 ESR2 (0.37) ESR2ESR1CYP2C9CYP3A4
SCHEMBL6043554 0.76 ESR2 (0.36) ESR2ESR1TDP1CA12CA1
SCHEMBL6043559 0.76 ESR2 (0.36) ESR2ESR1TDP1CA12CA1
SCHEMBL8337652 0.74 SLC18A3 (0.42) ESR2ESR1KDM1AMEN1KMT2A
SCHEMBL6954522 0.72 ESR2 (0.35) ESR2ESR1TDP1CA12CA1
SCHEMBL6041814 0.71 ESR2 (0.42) ESR2ESR1KDM1A
SCHEMBL6041817 0.71 ESR2 (0.42) ESR2ESR1KDM1A
SCHEMBL6042485 0.71 FUCA1 (0.63) ESR2ESR1ALDH1A1
SCHEMBL6042482 0.71 FUCA1 (0.63) ESR2ESR1ALDH1A1
SCHEMBL7447584 0.71 FUCA1 (0.63) ESR2ESR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175400-B1 RENIN INHIBITORS HOFFMANN LA ROCHE (CH) 2011-06-15 EP disclosed