SCHEMBL12600751

SCHEMBL12600751

CC(C)(C)[C@@H](CN1C(=O)c2ccccc2S1(=O)=O)NC=O

nearest known ligand 0.52

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CA12 O43570 13/20 0.52
CA9 Q16790 12/20 0.52
CA2 P00918 4/20 0.50
KMT2A Q03164 2/20 0.49
TDP1 Q9NUW8 1/20 0.49
ELANE P08246 1/20 0.49
KDM4E B2RXH2 1/20 0.48
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPT P10636 1/20 0.46
HPGD P15428 1/20 0.46
TSHR P16473 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
CA1 P00915 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12601260 0.86 CA12 (0.56) CA12CA9CA2KMT2ATDP1
SCHEMBL13632922 0.86 CA12 (0.56) CA12CA9CA2KMT2ATDP1
SCHEMBL8282041 0.78 TPSAB1 (0.54) CA12CA9CA2KMT2ATDP1
SCHEMBL13622671 0.78 TPSAB1 (0.54) CA12CA9CA2KMT2ATDP1
SCHEMBL8282960 0.78 CA12 (0.59) CA12CA9CA2KMT2ATDP1
SCHEMBL26232554 0.75 CA12 (0.68) CA12CA9CA2KMT2AELANE
SCHEMBL18026643 0.72 CA12 (0.68) CA12CA9CA2KMT2ATDP1
SCHEMBL8970514 0.70 CA12 (0.65) CA12CA9CA2ELANEALDH1A1
SCHEMBL1101896 0.70 CA12 (1.00) CA12CA9CA2ELANEALDH1A1
SCHEMBL30834902 0.70 CA12 (1.00) CA12CA9CA2ELANEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730142-B1 NOVEL KETOAMIDES WITH CYCLIC P4'S AS INHIBITORS OF NS3 SERINE PROTEASE OF HEPATITIS C VIRUS SCHERING CORP (US) 2011-06-29 EP disclosed