SCHEMBL12640604

SCHEMBL12640604

CCO[C@@H](C)c1ccc(CNC(=O)c2ccc(OCC(F)(F)F)nc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 12/20 0.55
CYP2C9 P11712 1/20 0.55
CYP2C19 P33261 1/20 0.55
CYP2J2 P51589 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.48
DGAT1 O75907 2/20 0.44
PPARG P37231 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
KCNH2 Q12809 1/20 0.42
SCN5A Q14524 1/20 0.42
SCN9A Q15858 1/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13876156 0.79 EPHX2 (0.81) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL13702303 0.78 L3MBTL1 (0.65) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL4189504 0.77 EPHX2 (0.82) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL13702153 0.75 L3MBTL1 (0.65) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL4178518 0.75 EPHX2 (0.73) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL15350981 0.74 EPHX2 (0.55) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL31498883 0.73 L3MBTL1 (0.65) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL15351096 0.73 EPHX2 (0.59) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL27931725 0.73 L3MBTL1 (0.54) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1
SCHEMBL13702416 0.73 L3MBTL1 (0.68) EPHX2CYP2C9CYP2C19CYP2J2L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011076678-A1 SUBSTITUTED BENZAMIDE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2011-06-30 WO disclosed