SCHEMBL12647751

SCHEMBL12647751

Brc1ccc2cc(-c3cnc[nH]3)ccc2c1

nearest known ligand 0.70

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.70
CYP11B2 P19099 2/20 0.70
IDO1 P14902 8/20 0.58
ASIC3 Q9UHC3 2/20 0.49
POLB P06746 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
CYP3A4 P08684 4/20 0.47
LTA4H P09960 1/20 0.46
CYP2D6 P10635 2/20 0.43
CYP2E1 P05181 1/20 0.43
CYP2A6 P11509 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2B6 P20813 1/20 0.43
CYP2C19 P33261 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26265591 0.89 CYP11B1 (0.85) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL20054668 0.84 CYP11B1 (0.77) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL26260218 0.83 CYP11B1 (0.82) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL2369049 0.82 CYP11B1 (1.00) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL205481 0.81 IDO1 (0.64) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL12647442 0.79 CYP11B1 (0.70) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL1502406 0.79 IDO1 (0.64) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL12647870 0.76 CYP11B1 (0.64) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL12647819 0.74 CYP11B1 (0.62) CYP11B1CYP11B2IDO1ASIC3POLB
SCHEMBL19792175 0.74 IDO1 (0.52) CYP11B1CYP11B2IDO1ASIC3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2499115-B1 PROCESS FOR PREPARING HEPATITIS C VIRUS INHIBITORS BRISTOL MYERS SQUIBB HOLDINGS IRELAND (CH) 2016-07-27 EP disclosed
WO-2011059887-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed
WO-2011059850-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-05-19 WO disclosed
WO-2011054834-A1 BENZIMIDAZOLE-IMIDAZOLE DERIVATIVES TIBOTEC PHARMACEUTICALS (IE) 2011-05-12 WO disclosed