SCHEMBL19792175

SCHEMBL19792175

FC1(F)c2cc(Br)ccc2-c2ccc(-c3cnc[nH]3)cc21

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 10/20 0.52
POLB P06746 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
CYP11B1 P15538 1/20 0.43
CYP11B2 P19099 1/20 0.43
ASIC3 Q9UHC3 2/20 0.41
SCN9A Q15858 1/20 0.39
CYP3A4 P08684 2/20 0.39
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
CYP2E1 P05181 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2A6 P11509 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2B6 P20813 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL206283 0.74 PDK2 (0.48) CYP2A6
SCHEMBL29540403 0.74 PDK2 (0.48) CYP2A6
SCHEMBL12647751 0.74 CYP11B1 (0.70) IDO1POLBSMN1; SMN2CYP11B1CYP11B2
SCHEMBL205481 0.73 IDO1 (0.64) IDO1POLBSMN1; SMN2CYP11B1CYP11B2
SCHEMBL21669605 0.71 IDO1 (0.63) IDO1POLBSMN1; SMN2CYP11B1CYP11B2
SCHEMBL13231061 0.71 PDK2 (0.46) MAPTCYP2A6
SCHEMBL1502406 0.71 IDO1 (0.64) IDO1POLBSMN1; SMN2CYP11B1CYP11B2
SCHEMBL1901766 0.69 IDO1 (1.00) IDO1POLBSMN1; SMN2ASIC3MAPT
SCHEMBL18829568 0.67 MAPK13 (0.40) SCN9A
SCHEMBL19764175 0.67 PDK2 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3272747-A1 METHOD OF PREPARATION FOR LEDIPASVIR AND DERIVATIVE THEREOF, AND INTERMEDIATE COMPOUND FOR PREPARATION OF LEDIPASVIR Shanghai Forefront Pharmceutical Co., Ltd (CN) 2018-01-24 EP disclosed