SCHEMBL12652103

SCHEMBL12652103

NS(=O)(=O)c1cc(F)cc(CNc2nc(NC3(C(F)(F)F)CC3)c3nc(C4CC4)ccc3n2)c1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.34
PTGS2 P35354 1/20 0.33
NTRK1 P04629 6/20 0.32
IKBKE Q14164 1/20 0.32
TBK1 Q9UHD2 1/20 0.32
CA1 P00915 4/20 0.31
CA2 P00918 4/20 0.31
CA9 Q16790 4/20 0.31
ADORA2A P29274 1/20 0.31
ADORA2B P29275 1/20 0.31
ADORA1 P30542 1/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30
PDE5A O76074 1/20 0.30
VCP P55072 1/20 0.30
PTK2 Q05397 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12652025 0.91 MAPK1 (0.34) MAPK1PTGS2NTRK1IKBKETBK1
SCHEMBL12652027 0.91 PTGS2 (0.34) PTGS2NTRK1IKBKETBK1CA1
SCHEMBL12651820 0.89 CA1 (0.43) PTGS2IKBKETBK1CA1CA2
SCHEMBL1791780 0.87 PTGS2 (0.38) PTGS2NTRK1CA2CA9ADORA2A
SCHEMBL1792358 0.85 NTRK1 (0.31) NTRK1
SCHEMBL1790384 0.84 NTRK1 (0.35) MAPK1PTGS2NTRK1PTK2
SCHEMBL1792271 0.81 PTGS2 (0.34) MAPK1PTGS2NTRK1PTK2
SCHEMBL1792081 0.80 TP53 (0.39) MAPK1PTGS2NTRK1CA1CA2
SCHEMBL1789966 0.80 PTGS2 (0.39) PTGS2ADORA2AMAPT
SCHEMBL1789942 0.80 PTGS2 (0.39) PTGS2CA1CA2CA9ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110123493-A1 2,4,6-TRISUBSTITUTED PYRIDO(3,2-d) PYRIMIDINES USEFUL FOR TREATING VIRAL INFECTIONS GILEAD SCIENCES, INC. (US) 2011-05-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110123493-A1 2,4,6-TRISUBSTITUTED PYRIDO(3,2-d) PYRIMIDINES USEFUL FOR TREATING VIRAL INFECTIONS PNPO, CYP2S1, DPYD MAPK1 2045/4885PTGS2 491/4885NTRK1 4157/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.