SCHEMBL12655873

SCHEMBL12655873

COc1ccc(CN2CCN(C(=O)Nc3ccc(O)cc3)CC2)cc1

nearest known ligand 0.80

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FAAH O00519 11/20 0.80
CA12 O43570 1/20 0.71
CA2 P00918 1/20 0.71
CA9 Q16790 1/20 0.71
MAPT P10636 1/20 0.68
PRKAB2 O43741 3/20 0.67
PRKAG1 P54619 3/20 0.67
PRKAA2 P54646 3/20 0.67
PRKAA1 Q13131 3/20 0.67
PRKAG3 Q9UGI9 3/20 0.67
PRKAG2 Q9UGJ0 3/20 0.67
PRKAB1 Q9Y478 3/20 0.67
POLB P06746 1/20 0.62
ALDH1A1 P00352 1/20 0.62
SMN1; SMN2 Q16637 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10839085 0.89 FAAH (0.91) FAAHCA12CA2CA9MAPT
SCHEMBL3606934 0.89 FAAH (1.00) FAAHMAPT
SCHEMBL12655875 0.86 FAAH (0.79) FAAHCA12CA2CA9MAPT
SCHEMBL12655878 0.85 FAAH (0.78) FAAHCA12CA2CA9MAPT
SCHEMBL13545510 0.84 FAAH (1.00) FAAHMAPTPRKAB2PRKAG1PRKAA2
SCHEMBL3592114 0.83 CA12 (0.90) FAAHCA12CA2CA9MAPT
SCHEMBL12655542 0.83 CA12 (1.00) FAAHCA12CA2CA9MAPT
SCHEMBL28869329 0.83 MAPT (1.00) FAAHCA12CA2CA9MAPT
SCHEMBL20236190 0.82 MAPT (0.80) FAAHMAPTPOLBSMN1; SMN2
SCHEMBL12655537 0.81 FAAH (0.80) FAAHCA12CA2CA9MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011060396-A1 ALIPHATIC AMINES BASED HETEROCYCLES USEFUL AS HIV ENTRY BLOCKERS SCHERING CORPORATION (US) 2011-05-19 WO disclosed