SCHEMBL12656128

SCHEMBL12656128

COc1ccc(S(=O)(=O)c2cn(-c3ccc4c(c3)B(O)OC4)c3ccccc23)cc1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.47
CA2 P00918 10/20 0.47
CA9 Q16790 9/20 0.47
CA4 P22748 8/20 0.47
CA7 P43166 8/20 0.47
PDE4A P27815 1/20 0.43
PDE4B Q07343 1/20 0.43
PDE4C Q08493 1/20 0.43
PDE4D Q08499 1/20 0.43
HTR6 P50406 1/20 0.38
TP53 P04637 1/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12656417 0.82 CA1 (0.48) CA1CA2CA9CA4CA7
SCHEMBL12656272 0.80 CA1 (0.48) CA1CA2CA9CA4CA7
SCHEMBL596472 0.77 PDE4A (0.58) CA1CA2CA9CA4CA7
SCHEMBL5583215 0.77 PDE4A (0.58) CA1CA2CA9CA4CA7
SCHEMBL2404339 0.71 CA1 (0.63) CA1CA2CA9CA4PDE4A
SCHEMBL595797 0.70 CA1 (0.50) CA1CA2CA9CA4CA7
SCHEMBL595739 0.70 CA1 (0.50) CA1CA2CA9CA4CA7
SCHEMBL12656464 0.69 CA1 (0.46) CA1CA2CA9CA4CA7
SCHEMBL28144965 0.69 NR4A2 (0.46) CA1CA2CA9HTR6TP53
SCHEMBL12656533 0.69 CA1 (0.43) CA1CA2CA9CA4CA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063293-A1 BORON-CONTAINING SMALL MOLECULES AS ANTIHELMINTH AGENTS ANACOR PHARMACEUTICALS, INC. (US) 2011-05-26 WO disclosed