SCHEMBL12656272

SCHEMBL12656272

COc1ccc(Sc2cn(-c3ccc4c(c3)B(O)OC4)c3ccccc23)cc1

nearest known ligand 0.48

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CA1 P00915 10/20 0.48
CA2 P00918 10/20 0.48
CA4 P22748 9/20 0.48
CA7 P43166 9/20 0.48
CA9 Q16790 9/20 0.48
PDE4A P27815 1/20 0.41
PDE4B Q07343 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL596135 0.90 CA1 (0.45) CA1CA2CA4CA7CA9
SCHEMBL595797 0.89 CA1 (0.50) CA1CA2CA4CA7CA9
SCHEMBL12656424 0.88 CA1 (0.43) CA1CA2CA4CA7CA9
SCHEMBL12656460 0.87 CA1 (0.43) CA1CA2CA4CA7CA9
SCHEMBL12656535 0.87 CA1 (0.46) CA1CA2CA4CA7CA9
SCHEMBL12656464 0.87 CA1 (0.46) CA1CA2CA4CA7CA9
SCHEMBL12656271 0.87 CA1 (0.43) CA1CA2CA4CA7CA9
SCHEMBL12656127 0.84 CA1 (0.41) CA1CA2CA4CA7CA9
SCHEMBL12656427 0.83 CA1 (0.51) CA1CA2CA4CA7CA9
SCHEMBL12656534 0.82 CA1 (0.43) CA1CA2CA4CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063293-A1 BORON-CONTAINING SMALL MOLECULES AS ANTIHELMINTH AGENTS ANACOR PHARMACEUTICALS, INC. (US) 2011-05-26 WO disclosed