SCHEMBL12656336

SCHEMBL12656336

CCN1CCc2cc(Cl)c(Cl)cc21

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 8/20 0.49
HTR2C P28335 8/20 0.49
HTR2B P41595 8/20 0.49
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
NOTUM Q6P988 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
PNMT P11086 1/20 0.37
ACHE P22303 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
NFKB1 P19838 1/20 0.34
HIF1A Q16665 1/20 0.34
HRH3 Q9Y5N1 2/20 0.34
HSP90AA1 P07900 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4050281 0.87 HDAC1 (0.49) HTR2AHTR2CHTR2BHDAC1HDAC6
SCHEMBL14473195 0.86 HTR2A (0.67) HTR2AHTR2CHTR2BHDAC1HDAC6
SCHEMBL12735193 0.85 HTR2A (0.47) HTR2AHTR2CHTR2BHDAC1HDAC6
SCHEMBL28942333 0.78 HTR2A (0.65) HTR2AHTR2CHTR2BHDAC1HDAC6
SCHEMBL29803467 0.77 NOTUM (0.40) HTR2AHTR2CHTR2BNOTUMACHE
SCHEMBL107921 0.77 NOTUM (0.40) HTR2AHTR2CHTR2BNOTUMACHE
Ammonia Solution, Strong SCHEMBL906017 0.77 HTR2A (0.63) HTR2AHTR2CHTR2BHDAC1HDAC6
SCHEMBL20651648 0.76 HDAC1 (0.36) HTR2AHTR2CHTR2BHDAC1HDAC6
SCHEMBL21469192 0.76 SMN1; SMN2 (0.48) CYP1A2CYP3A4CYP2D6
Bromide SCHEMBL9480957 0.76 DRD2 (0.40) HTR2AHTR2CHTR2BNOTUMACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2316829-A1 Heterocyclic derivatives as modulators of ion channels Vertex Pharmaceuticals Incorporated (US) 2011-05-04 EP disclosed