SCHEMBL12658662

SCHEMBL12658662

Cn1ccc(NC(=O)NCc2cccc(O)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 1/20 0.49
MAPT P10636 2/20 0.48
MTOR P42345 2/20 0.45
ROCK2 O75116 4/20 0.45
ROCK1 Q13464 3/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
SGK1 O00141 1/20 0.43
AKT1 P31749 1/20 0.43
GSK3B P49841 1/20 0.43
LIMK1 P53667 1/20 0.43
TNK2 Q07912 1/20 0.43
DMPK Q09013 1/20 0.43
MYLK Q15746 1/20 0.43
CDC42BPA Q5VT25 1/20 0.43
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
L3MBTL1 Q9Y468 2/20 0.43
USP2 O75604 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL357618 0.80 TSHR (0.53) HIF1AMAPTROCK2ROCK1SMN1; SMN2
SCHEMBL356085 0.78 ROCK2 (0.46) HIF1AMAPTROCK2ROCK1SMN1; SMN2
SCHEMBL13984317 0.76 ERCC1 (0.60) HIF1AMAPTMTORROCK2ROCK1
SCHEMBL14289839 0.74 CYP1A2 (0.53) HIF1AMAPTROCK2ROCK1SGK1
SCHEMBL25709720 0.73 MTOR (0.62) HIF1AMAPTMTORROCK2ROCK1
SCHEMBL359215 0.72 ROCK2 (0.46) HIF1AMAPTROCK2ROCK1SMN1; SMN2
SCHEMBL22026435 0.71 CYP1A2 (0.62) HIF1AMAPTROCK2ROCK1KMT2A
SCHEMBL358332 0.71 CYP1A2 (0.61) HIF1AMAPTROCK2ROCK1KMT2A
SCHEMBL31724652 0.71 CYP1A2 (0.56) HIF1AMAPTROCK2ROCK1KMT2A
SCHEMBL5725833 0.71 CYP1A2 (0.56) HIF1AMAPTROCK2ROCK1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2322525-A1 Purine derivatives for use as adenosin A2A receptor agonists Novartis AG (CH) 2011-05-18 EP disclosed