SCHEMBL12662829

SCHEMBL12662829

C=Cc1cc(C)cc(OC)c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 5/20 0.48
CYP1B1 Q16678 5/20 0.48
TP53 P04637 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
ALDH1A1 P00352 1/20 0.42
NQO2 P16083 4/20 0.41
CYP1A2 P05177 3/20 0.41
ABL1 P00519 3/20 0.41
BCR P11274 3/20 0.41
ESR1 P03372 2/20 0.41
TTR P02766 2/20 0.41
ABCB1 P08183 2/20 0.41
ALOX5 P09917 2/20 0.41
CYP19A1 P11511 2/20 0.41
PTGS2 P35354 2/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
AHR P35869 1/20 0.41
TUBA1B P68363 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31618743 1.00 CYP1A1 (0.48) CYP1A1CYP1B1TP53TDP1ALDH1A1
SCHEMBL2017917 0.86 CYP1A1 (0.64) CYP1A1CYP1B1ALDH1A1NQO2CYP1A2
SCHEMBL25195786 0.86 CYP1A1 (0.56) CYP1A1CYP1B1ALDH1A1NQO2CYP1A2
SCHEMBL4455795 0.84 TDP1 (0.45) CYP1A1CYP1B1TP53TDP1ALDH1A1
Methoxymethane SCHEMBL28654805 0.84 CYP1A1 (0.61) CYP1A1CYP1B1ALDH1A1NQO2CYP1A2
Methoxymethane SCHEMBL28663826 0.81 TDP1 (0.50) TP53TDP1ALDH1A1ACHERELA
SCHEMBL16362233 0.80 CYP1A1 (0.77) CYP1A1CYP1B1NQO2CYP1A2ABL1
SCHEMBL9928608 0.78 CYP1A1 (0.58) CYP1A1CYP1B1TP53ALDH1A1NQO2
SCHEMBL16958243 0.78 CYP1A1 (0.48) CYP1A1CYP1B1TP53ALDH1A1NQO2
SCHEMBL29951799 0.78 ALDH1A1 (0.50) CYP1A1CYP1B1TDP1ALDH1A1NQO2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11661397-B2 1,4-disubstituted imidazole derivative Sumitomo Pharma Co., Ltd. (JP) 2023-05-30 US disclosed
CN-108640839-B Intermolecular 1, 2-dialkylation reaction method of olefin compound under photo-oxidation-reduction/iron (II) catalytic system 南昌航空大学 2021-01-05 CN disclosed
US-9828362-B2 1,4-disubstituted imidazole derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2017-11-28 US disclosed
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2017-06-15 US disclosed
US-9643946-B2 Tricyclic compound and use thereof SK CHEMICALS CO., LTD. (KR) 2017-05-09 US disclosed
US-9493436-B2 Tyrosine phosphatase inhibitors and uses thereof to modulate the activity of enzymes involved in the pathology of Mycobacterium tuberculosis INDIANA UNIVERSITY RESEARCH AND TECHNOLOGY CORPORATION (US) 2016-11-15 US disclosed
EP-2900645-A1 3-PHENYLISOXAZOLIN DERIVATIVES WITH HERBICIDAL ACTION Bayer CropScience AG (DE) 2015-08-05 EP disclosed
EP-2125748-B1 ACYLAMINOPYRAZOLES AS FGFR INHIBITORS ASTRAZENECA AB (SE) 2011-05-25 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170166552-A1 1,4-DISUBSTITUTED IMIDAZOLE DERIVATIVE NR4A3, NR0B1, NR2C2 CYP1A1 389/4885CYP1B1 611/4885TP53 247/4885
US-11661397-B2 1,4-disubstituted imidazole derivative NR4A3, NR0B1, NR2C2 CYP1A1 389/4885CYP1B1 611/4885TP53 247/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.