SCHEMBL12663929

SCHEMBL12663929

COc1cc(C2CC2)c2ccccc2c1-n1c(N)nnc1SCC(=O)Nc1ccc(S(N)(=O)=O)cc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.44
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 1/20 0.43
EGFR P00533 1/20 0.43
ERBB2 P04626 1/20 0.43
MAPK1 P28482 1/20 0.42
CA1 P00915 4/20 0.42
CA2 P00918 4/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
SLC22A12 Q96S37 1/20 0.41
SLC2A9 Q9NRM0 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
POLB P06746 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12628980 0.92 SLC22A12 (0.49) ALDH1A1MEN1KMT2ANPC1EGFR
SCHEMBL12011515 0.91 EGFR (0.44) ALDH1A1MEN1KMT2AEGFRERBB2
SCHEMBL247372 0.86 SLC22A12 (0.54) EGFRERBB2CA1CA2CA9
SCHEMBL12011401 0.83 CA1 (0.46) ALDH1A1NPC1EGFRERBB2CA1
SCHEMBL843082 0.83 SLC22A12 (0.51) ALDH1A1MEN1KMT2AEGFRERBB2
SCHEMBL1719515 0.82 EGFR (0.43) ALDH1A1MEN1KMT2AEGFRERBB2
SCHEMBL3435532 0.81 SLC22A12 (0.54) EGFRERBB2CA1CA2CA9
SCHEMBL13825281 0.79 SLC22A12 (0.54) EGFRERBB2CA1CA2CA9
SCHEMBL30601618 0.79 SLC22A12 (0.66) EGFRERBB2CA1CA2CA12
SCHEMBL248867 0.79 SLC22A12 (0.66) EGFRERBB2CA1CA2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7947721-B2 able to inhibit various mutated RTs, including K103N, Y181C and Y188L Ardes Biosciences Inc. (US) 2011-05-24 US disclosed