SCHEMBL12683258

SCHEMBL12683258

CC(C)c1nc2ccc(F)cc2n1-c1ccncc1

nearest known ligand 0.52

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 4/20 0.52
PIK3CD O00329 7/20 0.45
PIK3R1 P27986 7/20 0.45
PIK3CB P42338 7/20 0.45
PIK3CG P48736 7/20 0.45
PIK3CA P42336 6/20 0.45
CYP11B1 P15538 4/20 0.42
CYP11B2 P19099 4/20 0.42
CYP1A2 P05177 1/20 0.41
CRBN Q96SW2 1/20 0.40
GSR P00390 1/20 0.39
AAK1 Q2M2I8 1/20 0.36
AOC3 Q16853 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11901355 0.89 PIK3CD (0.46) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
SCHEMBL12683083 0.83 PIK3CD (0.57) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
SCHEMBL11901816 0.78 PIK3CD (0.54) PIK3CDPIK3R1PIK3CBPIK3CGPIK3CA
SCHEMBL2503207 0.78 PIK3CD (0.54) PIK3CDPIK3R1PIK3CBPIK3CGPIK3CA
SCHEMBL11901385 0.77 PIK3CD (0.42) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
SCHEMBL12473152 0.76 PIK3CD (0.55) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
SCHEMBL2505813 0.76 PIK3CD (0.55) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
Hydrochloric Acid SCHEMBL11901325 0.75 PIK3CD (0.54) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
Hydrochloric Acid SCHEMBL12473126 0.75 PIK3CD (0.54) PDE10APIK3CDPIK3R1PIK3CBPIK3CG
SCHEMBL2509454 0.74 PIK3CD (0.54) PIK3CDPIK3R1PIK3CBPIK3CGPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012107465-A1 HETEROCYCLIC COMPOUNDS AS PI3 KINASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2012-08-16 WO disclosed