SCHEMBL12700558

SCHEMBL12700558

COCc1cccc(-c2ocnc2CN2CCNC3(CCN(c4nc(C)cc(N)n4)CC3)C2=O)c1

nearest known ligand 0.38

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.38
HCRTR2 O43614 16/20 0.38
GRM5 P41594 1/20 0.34
MTOR P42345 1/20 0.33
CES2 O00748 1/20 0.32
PIK3CA P42336 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9949057 0.95 HCRTR1 (0.41) HCRTR1HCRTR2GRM5CES2
SCHEMBL9948745 0.92 HCRTR1 (0.38) HCRTR1HCRTR2GRM5CES2
SCHEMBL9949076 0.90 HCRTR1 (0.38) HCRTR1HCRTR2GRM5CES2
SCHEMBL12700557 0.90 HCRTR1 (0.40) HCRTR1HCRTR2CES2
SCHEMBL12700478 0.89 HCRTR1 (0.39) HCRTR1HCRTR2MTORCES2PIK3CA
SCHEMBL9948877 0.85 HCRTR1 (0.44) HCRTR1HCRTR2CES2
SCHEMBL9949015 0.84 HCRTR1 (0.43) HCRTR1HCRTR2MTORCES2PIK3CA
SCHEMBL9948925 0.82 SLC6A2 (0.42) HCRTR1HCRTR2CES2
SCHEMBL2131622 0.82 HCRTR1 (0.57) HCRTR1HCRTR2
SCHEMBL9948794 0.81 HCRTR1 (0.39) HCRTR1HCRTR2CES2PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012101487-A1 DI/TRI-AZA-SPIRO-C9-C11ALKANES NOVARTIS AG (CH) 2012-08-02 WO disclosed