SCHEMBL12733692

SCHEMBL12733692

CCC(C)C1(C)CC2(CCCNC2)C1

nearest known ligand 0.31

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
TSHR P16473 2/20 0.31
USP2 O75604 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15533767 0.82
SCHEMBL15533908 0.74 TSHR (0.32) TSHR
SCHEMBL10287479 0.73 CYP3A4 (0.36) CYP3A4CYP2D6TSHRUSP2ALDH1A1
SCHEMBL2755099 0.72 CYP2D6 (0.34) CYP3A4CYP2D6TSHRUSP2ALDH1A1
SCHEMBL15533181 0.71
SCHEMBL24536722 0.70 ALDH1A1 (0.34) CYP3A4CYP2D6TSHRUSP2ALDH1A1
SCHEMBL20329284 0.70 TSHR (0.35) TSHR
SCHEMBL21217092 0.69 CYP2D6 (0.42) CYP3A4CYP2D6TSHRUSP2ALDH1A1
SCHEMBL22279859 0.69 CYP3A4 (0.36) CYP3A4CYP2D6TSHRUSP2ALDH1A1
SCHEMBL165883 0.67 CYP2D6 (0.42) CYP3A4CYP2D6TSHRUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110082135-A1 INHIBITORS OF AKT ACTIVITY MERCK SHARP & DOHME LLC 2011-04-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110082135-A1 INHIBITORS OF AKT ACTIVITY PIK3CA, AKT1S1, AKT1 CYP3A4 3065/4885CYP2D6 3866/4885TSHR 3128/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.