SCHEMBL1274041

SCHEMBL1274041

C=Cc1ccc2nc(-c3ccccc3)cc(O[C@H]3CN(C(=O)OC(C)(C)C)[C@](C)(C(=O)O)C3)c2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 4/20 0.34
HTR3E A5X5Y0 1/20 0.33
HTR3B O95264 1/20 0.33
HTR3A P46098 1/20 0.33
HTR3D Q70Z44 1/20 0.33
HTR3C Q8WXA8 1/20 0.33
UCHL1 P09936 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
BACE1 P56817 3/20 0.31
USP30 Q70CQ3 3/20 0.31
ACACA Q13085 2/20 0.31
GBA1 P04062 1/20 0.31
ADAM17 P78536 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
CKS1B P61024 1/20 0.31
SKP1 P63208 1/20 0.31
SKP2 Q13309 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1072632 0.89 SMN1; SMN2 (0.36) ACACBUCHL1KDM4EMEN1KMT2A
SCHEMBL1273640 0.88 RXFP1 (0.42) ACACBHTR3EHTR3BHTR3AHTR3D
SCHEMBL1274307 0.86 ACACB (0.34) ACACBHTR3EHTR3BHTR3AHTR3D
SCHEMBL1072461 0.83 SMN1; SMN2 (0.35) ACACBUCHL1KDM4EMEN1KMT2A
SCHEMBL8253556 0.79 UCHL1 (0.45) ACACBHTR3EHTR3BHTR3AHTR3D
SCHEMBL1071232 0.79 PIK3CD (0.33)
SCHEMBL2428718 0.79 CYP3A4 (0.32)
Hydrochloric Acid SCHEMBL1071700 0.78 PIK3CD (0.33)
SCHEMBL1072152 0.75 MEN1 (0.41) ACACBMEN1KMT2ABACE1ACACA
SCHEMBL1083306 0.75 MEN1 (0.41) ACACBMEN1KMT2ABACE1ACACA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879797-B2 HCV NS3 protease inhibitors MERCK SHARP & DOHME CORP. (US) 2011-02-01 US disclosed