SCHEMBL12774151

SCHEMBL12774151

CCOC(=O)OC(C)OC(=O)CCCN1CCC(N2CCN(C)CC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 2/20 0.36
HTR4 Q13639 2/20 0.35
TDP1 Q9NUW8 1/20 0.35
MGLL Q99685 1/20 0.35
CHRM1 P11229 1/20 0.34
SMN1; SMN2 Q16637 5/20 0.34
PAOX Q6QHF9 1/20 0.32
L3MBTL3 Q96JM7 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
GAA P10253 1/20 0.32
ALOX12 P18054 1/20 0.32
ACHE P22303 1/20 0.31
MAPK1 P28482 1/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
RAD52 P43351 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12774140 0.93 TP53 (0.42) TP53TDP1MGLLCHRM1SMN1; SMN2
SCHEMBL12774086 0.87 CYP1A2 (0.37) TP53TDP1CHRM1SMN1; SMN2L3MBTL3
SCHEMBL12774129 0.84 HTR4 (0.42) TP53HTR4TDP1CHRM1SMN1; SMN2
SCHEMBL12774050 0.83 CYP1A2 (0.40) TP53TDP1CHRM1SMN1; SMN2L3MBTL3
SCHEMBL13601528 0.81 TP53 (0.43) TP53MGLLSMN1; SMN2PAOXALDH1A1
SCHEMBL13601439 0.77 POLB (0.43) TP53MGLLSMN1; SMN2L3MBTL1HRH3
SCHEMBL12881438 0.77 TP53 (0.47) TP53TDP1CHRM1SMN1; SMN2GAA
SCHEMBL12774197 0.76 CHRM1 (0.38) TP53TDP1CHRM1SMN1; SMN2L3MBTL3
SCHEMBL12774124 0.76 HRH3 (0.42) TP53SMN1; SMN2HRH3ACHEMAPK1
SCHEMBL12774104 0.76 TP53 (0.49) TP53TDP1SMN1; SMN2L3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7897603-B2 Selected CGRP-antagonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-03-01 US disclosed