SCHEMBL12801331

SCHEMBL12801331

COc1cc(NC(=O)NC2CCN(C)CC2)cc(Nc2nccc(-c3ccc(OC)c(N)c3)n2)c1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCNC P24863 3/20 0.48
CDK8 P49336 3/20 0.48
GSK3B P49841 1/20 0.47
ZAP70 P43403 5/20 0.46
JAK2 O60674 3/20 0.44
JAK3 P52333 1/20 0.42
CDK5 Q00535 1/20 0.42
SYK P43405 2/20 0.42
IKBKB O14920 2/20 0.42
BRD4 O60885 1/20 0.41
CCNA2 P20248 1/20 0.41
CDK2 P24941 1/20 0.41
CCNA1 P78396 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12521964 0.92 CCNC (0.47) CCNCCDK8GSK3BZAP70JAK2
SCHEMBL12801322 0.92 GSK3B (0.49) CCNCCDK8GSK3BJAK2CDK5
SCHEMBL12801341 0.91 GSK3B (0.49) CCNCCDK8GSK3BZAP70JAK2
SCHEMBL12275308 0.89 CCNC (0.46) CCNCCDK8GSK3BZAP70
SCHEMBL12801368 0.84 GSK3B (0.43) CCNCCDK8GSK3BZAP70JAK2
SCHEMBL12801676 0.83 AURKB (0.55) JAK2JAK3CDK5IKBKB
SCHEMBL12801697 0.83 ABL1 (0.50) JAK2CDK5CDK2
SCHEMBL12801695 0.83 IKBKB (0.52) GSK3BJAK2JAK3CDK5IKBKB
SCHEMBL12801280 0.82 IKBKB (0.58) ZAP70JAK2JAK3CDK5IKBKB
SCHEMBL12801123 0.82 PDPK1 (0.49) ZAP70JAK2JAK3CDK5SYK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed