SCHEMBL12801697

SCHEMBL12801697

COc1ccc(-c2ccnc(Nc3cccc(NC(=O)NC4CCCC4)c3)n2)cc1N

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 5/20 0.50
BCR P11274 5/20 0.50
PDGFRB P09619 2/20 0.50
PDGFRA P16234 2/20 0.50
EGFR P00533 2/20 0.50
PRKCA P17252 1/20 0.50
SRC P12931 1/20 0.50
CDK5 Q00535 1/20 0.49
PDPK1 O15530 2/20 0.48
NPC1 O15118 1/20 0.48
RAB9A P51151 1/20 0.48
KDR P35968 2/20 0.48
JAK2 O60674 2/20 0.47
FLT3 P36888 1/20 0.47
AURKB Q96GD4 1/20 0.46
CAMKK1 Q8N5S9 1/20 0.45
CAMKK2 Q96RR4 1/20 0.45
ERBB2 P04626 1/20 0.45
MET P08581 1/20 0.45
MERTK Q12866 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801676 0.92 AURKB (0.55) PDGFRACDK5NPC1RAB9AKDR
SCHEMBL12801322 0.91 GSK3B (0.49) ABL1BCRPDGFRBPDGFRAEGFR
SCHEMBL12801341 0.90 GSK3B (0.49) PDGFRACDK5NPC1RAB9AKDR
SCHEMBL12274595 0.88 GSK3B (0.48) ABL1BCRPDGFRBPDGFRAEGFR
SCHEMBL12801304 0.85 ABL1 (0.58) ABL1BCRPDGFRBPDGFRAEGFR
SCHEMBL12801096 0.85 JAK2 (0.61) ABL1BCRPDGFRBPDGFRAEGFR
SCHEMBL12801331 0.83 CCNC (0.48) CDK5JAK2CDK2
SCHEMBL12522222 0.83 ABL1 (0.51) ABL1BCRPDGFRBPDGFRAEGFR
SCHEMBL12801324 0.83 PDPK1 (0.59) ABL1BCRPDGFRBPDGFRAEGFR
SCHEMBL12521964 0.82 CCNC (0.47) CDK5JAK2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed