SCHEMBL12801367

SCHEMBL12801367

C[C@H](O)C(=O)N1CCC(Oc2ccc(-c3ccnc(Nc4ccc(C(=O)N(C)CCN(C)C)cc4)n3)cc2N)CC1

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 12/20 0.45
JAK2 O60674 4/20 0.43
MYLK4 Q86YV6 2/20 0.43
STK17A Q9UEE5 2/20 0.43
NEK3 P51956 1/20 0.43
LIMK1 P53667 1/20 0.43
NEK5 Q6P3R8 1/20 0.43
JAK3 P52333 1/20 0.43
CDK2 P24941 3/20 0.41
CCNA2 P20248 1/20 0.41
CDK1 P06493 1/20 0.39
CDC7 O00311 1/20 0.39
CDK19 Q9BWU1 1/20 0.39
IKBKB O14920 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801379 0.90 CDC7 (0.51) TBK1JAK2MYLK4STK17ANEK3
SCHEMBL1667478 0.90 TBK1 (0.57) TBK1JAK2
SCHEMBL12800894 0.89 CDC7 (0.46) TBK1JAK2MYLK4STK17ANEK3
SCHEMBL12801598 0.88 TBK1 (0.48) TBK1JAK2MYLK4STK17ANEK3
SCHEMBL12801665 0.88 TBK1 (0.48) TBK1JAK2MYLK4STK17ANEK3
SCHEMBL12801538 0.85 TBK1 (0.53) TBK1JAK2MYLK4STK17ANEK3
SCHEMBL12801252 0.83 JAK2 (0.59) TBK1JAK2JAK3
SCHEMBL12801663 0.83 JAK2 (0.59) TBK1JAK2JAK3
SCHEMBL12801316 0.83 JAK2 (0.45) TBK1JAK2JAK3CDK2CCNA2
SCHEMBL12800954 0.82 JAK2 (0.52) TBK1JAK2STK17AJAK3CDK19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed