SCHEMBL128015

SCHEMBL128015

c1ccc(-c2cccc(-c3cc4ccccc4cn3)c2)cc1

nearest known ligand 0.78

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.54
RAB9A P51151 2/20 0.54
IDO1 P14902 1/20 0.53
TDO2 P48775 1/20 0.53
KMO O15229 2/20 0.47
CYP1A2 P05177 2/20 0.44
CYP2A6 P11509 1/20 0.44
PDPK1 O15530 1/20 0.44
KDM4E B2RXH2 2/20 0.44
TDP1 Q9NUW8 1/20 0.44
BTK Q06187 1/20 0.44
HSD17B1 P14061 1/20 0.41
HSD17B2 P37059 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21173250 0.92 NPC1 (0.58) NPC1RAB9AIDO1TDO2CYP1A2
SCHEMBL17413708 0.92 NPC1 (0.51) NPC1RAB9AIDO1TDO2KMO
SCHEMBL17343432 0.92 NPC1 (0.47) NPC1RAB9AIDO1TDO2KMO
SCHEMBL129816 0.90 NPC1 (0.56) NPC1RAB9AIDO1TDO2CYP1A2
SCHEMBL17944930 0.90 NPC1 (0.54) NPC1RAB9AIDO1TDO2KMO
SCHEMBL17367803 0.90 MEN1 (0.49) NPC1RAB9AIDO1TDO2KMO
SCHEMBL17343378 0.90 NPC1 (0.46) NPC1RAB9AIDO1TDO2KMO
SCHEMBL17944936 0.89 NPC1 (0.53) NPC1RAB9AIDO1TDO2KDM4E
SCHEMBL17944926 0.89 NPC1 (0.53) NPC1RAB9AIDO1TDO2KDM4E
SCHEMBL18858310 0.89 NPC1 (0.53) NPC1RAB9AIDO1TDO2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed
WO-2010127307-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2010-11-04 WO disclosed
WO-2010127307-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2010-11-04 WO disclosed
US-7429426-B2 Organometallic compounds for use in electroluminescent devices THE UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2008-09-30 US disclosed
US-7429426-B2 Organometallic compounds for use in electroluminescent devices THE UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2008-09-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059026-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L NPC1 866/4885RAB9A 1144/4885IDO1 588/4885
US-20140315939-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L NPC1 799/4885RAB9A 964/4885IDO1 864/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.