SCHEMBL12801543

SCHEMBL12801543

COc1ccc(-c2ccnc(Nc3ccc(N4CCOCC4)c(Cl)c3)n2)cc1N

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 6/20 0.67
JAK3 P52333 2/20 0.60
ZAP70 P43403 1/20 0.54
SMG1 Q96Q15 5/20 0.53
MTOR P42345 1/20 0.53
CDK2 P24941 3/20 0.51
CDK1 P06493 2/20 0.51
CAMK2D Q13557 1/20 0.51
KCNH2 Q12809 1/20 0.51
TNIK Q9UKE5 1/20 0.51
CCNT1 O60563 2/20 0.50
CDK9 P50750 2/20 0.50
MAPK8 P45983 1/20 0.49
MAPK9 P45984 1/20 0.49
MAPK10 P53779 1/20 0.49
IGF1R P08069 1/20 0.49
CCNA2 P20248 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12801124 0.88 JAK2 (0.54) JAK2JAK3SMG1CDK2CDK1
SCHEMBL12801653 0.88 JAK2 (0.85) JAK2JAK3ZAP70CDK2CDK1
SCHEMBL1670016 0.87 JAK2 (0.57) JAK2JAK3ZAP70SMG1MTOR
SCHEMBL27898071 0.85 JAK2 (0.59) JAK2JAK3ZAP70SMG1MTOR
SCHEMBL12801393 0.85 JAK2 (0.69) JAK2JAK3ZAP70SMG1MTOR
SCHEMBL12801232 0.85 JAK2 (0.61) JAK2JAK3ZAP70SMG1MTOR
SCHEMBL13588456 0.84 JAK2 (0.67) JAK2JAK3ZAP70SMG1MTOR
Hydrochloric Acid SCHEMBL4383810 0.83 JAK2 (0.66) JAK2JAK3ZAP70SMG1MTOR
SCHEMBL12801647 0.82 JAK2 (0.60) JAK2JAK3ZAP70SMG1MTOR
SCHEMBL8093455 0.81 JAK2 (0.61) JAK2JAK3ZAP70SMG1MTOR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed