SCHEMBL12801545

SCHEMBL12801545

N#Cc1cc(-c2ccnc(Nc3ccc(N4CCOCC4)cc3)n2)ccc1OC1CCN(S)CC1

nearest known ligand 0.67

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 19/20 0.67
JAK2 O60674 5/20 0.67
IKBKE Q14164 14/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29772697 0.93 TBK1 (0.76) TBK1JAK2IKBKE
SCHEMBL1667556 0.93 TBK1 (0.76) TBK1JAK2IKBKE
SCHEMBL1667172 0.92 TBK1 (0.69) TBK1JAK2IKBKE
SCHEMBL1667100 0.90 TBK1 (0.71) TBK1JAK2IKBKE
SCHEMBL1667187 0.90 TBK1 (0.64) TBK1JAK2IKBKE
SCHEMBL12274012 0.90 TBK1 (0.64) TBK1JAK2IKBKE
SCHEMBL12522280 0.90 TBK1 (0.64) TBK1JAK2IKBKE
SCHEMBL1667659 0.89 TBK1 (0.70) TBK1JAK2IKBKE
SCHEMBL12275053 0.89 TBK1 (0.63) TBK1JAK2IKBKE
SCHEMBL1667417 0.89 TBK1 (0.63) TBK1JAK2IKBKE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011046970-A1 AMINO - PYRIMIDINE COMPOUNDS AS INHIBITORS OF TBKL AND/OR IKK EPSILON MYREXIS, INC. (US) 2011-04-21 WO disclosed