SCHEMBL12808643

SCHEMBL12808643

CC1=C(NC(=O)CCc2ccc(-c3ccccc3)cc2)CCC1

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 12/20 0.58
FFAR1 O14842 1/20 0.49
MMP12 P39900 1/20 0.48
LTB4R Q15722 1/20 0.47
NAAA Q02083 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
CNR2 P34972 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4548322 0.84 HCAR2 (0.81) HCAR2
SCHEMBL4548317 0.83 HCAR2 (0.83) HCAR2FFAR1
SCHEMBL4548396 0.81 HCAR2 (0.55) HCAR2FFAR1MMP12NAAAMAPT
SCHEMBL10312490 0.79 HCAR2 (0.53) HCAR2FFAR1MMP12LTB4RNAAA
SCHEMBL4548327 0.75 HCAR2 (0.48) HCAR2FFAR1MMP12NAAA
SCHEMBL4548312 0.73 HCAR2 (0.77) HCAR2MAPT
SCHEMBL13356363 0.72 MAPT (0.80) MAPTHTT
SCHEMBL7046207 0.72 HDAC1 (0.79) FFAR1MMP12
SCHEMBL13781562 0.71 HCAR2 (0.58) HCAR2LTB4RMAPTHTT
SCHEMBL13781560 0.71 ALDH1A1 (0.56) HCAR2LTB4RMAPTHTTCNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1901731-B1 NIACIN RECEPTOR AGONISTS, COMPOSITIONS CONTAINING SUCH COMPOUNDS AND METHODS OF TREATMENT MERCK SHARP & DOHME (US) 2011-03-02 EP disclosed