SCHEMBL12811481

SCHEMBL12811481

CC(=O)N1Cc2nc(N)nc(N)c2C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.35
KDM4E B2RXH2 2/20 0.34
CYP1A2 P05177 2/20 0.34
ALDH1A1 P00352 1/20 0.34
HPGD P15428 1/20 0.34
CYP2C19 P33261 1/20 0.33
BPTF Q12830 1/20 0.33
P2RX7 Q99572 1/20 0.32
CHRM4 P08173 1/20 0.32
IKBKB O14920 1/20 0.32
MAP3K14 Q99558 1/20 0.32
PDPK1 O15530 1/20 0.32
HSP90AA1 P07900 3/20 0.31
HSP90AB1 P08238 3/20 0.31
MAP4K4 O95819 1/20 0.31
BAZ2B Q9UIF8 1/20 0.31
CASP6 P55212 1/20 0.30
GFER P55789 1/20 0.30
AURKA O14965 1/20 0.30
CCNA2 P20248 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3264107 0.76 HRH4 (0.41) CYP1A2
SCHEMBL20608495 0.71 CHRM4 (0.34) CYP1A2P2RX7CHRM4
SCHEMBL20618233 0.70 NOTUM (0.36) NOTUMCYP1A2ALDH1A1P2RX7CHRM4
SCHEMBL18343220 0.69 NOTUM (0.35) NOTUMCYP1A2CHRM4BAZ2BAURKA
SCHEMBL2923652 0.69 CCNA2 (0.38) NOTUMBAZ2BAURKACCNA2CDK2
SCHEMBL15189253 0.69 CYP2C19 (0.35) KDM4ECYP2C19
SCHEMBL13495928 0.68 KDM4E (0.40) KDM4ECYP1A2ALDH1A1HPGD
SCHEMBL23253676 0.68 CHRM4 (0.63) NOTUMKDM4ECYP1A2ALDH1A1HPGD
SCHEMBL3241010 0.68 P2RX7 (0.34) P2RX7HSP90AA1HSP90AB1
SCHEMBL1425313 0.66 MAPT (0.38) KDM4ECYP1A2ALDH1A1HPGDCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2118111-B1 2-AMIN0-5, 7-DIHYDR0-6H- PYRROLO [3, 4-D] PYRIMIDINE DERIVATIVES AS HSP-90 INHIBITORS FOR TREATING CANCER PFIZER (US) 2011-03-23 EP disclosed