SCHEMBL12820036

SCHEMBL12820036

NC(=O)c1ccc(-c2c3n(c4ccccc24)C(=O)CCC3)cc1N[C@H]1CC[C@H](O)CC1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 20/20 0.47
HSP90AB1 P08238 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12819874 0.94 HSP90AA1 (0.48) HSP90AA1HSP90AB1
SCHEMBL12819989 0.93 ROCK2 (0.40) HSP90AA1HSP90AB1
SCHEMBL12819609 0.93 HSP90AA1 (0.42) HSP90AA1HSP90AB1
SCHEMBL12819517 0.91 HSP90AA1 (0.46) HSP90AA1HSP90AB1
SCHEMBL12819508 0.90 HSP90AA1 (0.40) HSP90AA1HSP90AB1
SCHEMBL12819744 0.90 HSP90AA1 (0.43) HSP90AA1HSP90AB1
SCHEMBL12819928 0.90 HSP90AA1 (0.45) HSP90AA1HSP90AB1
SCHEMBL12819759 0.90 AURKA (0.39) HSP90AA1HSP90AB1
SCHEMBL12819858 0.89 HSP90AA1 (0.39) HSP90AA1HSP90AB1
SCHEMBL12819773 0.89 HSP90AA1 (0.42) HSP90AA1HSP90AB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012126084-A1 HSP-90 BINDING COMPOUNDS, COMPOSITIONS THEREOF, AND THEIR USE IΝ THE TREATMENT AND PREVENTION OF FUNGAL INFECTIONS PHARMASCIENCE INC. (CA) 2012-09-27 WO disclosed
WO-2011035417-A1 HSP-90 BINDING COMPOUNDS, COMPOSITIONS THEREOF, AND THEIR USE FN THE TREATMENT OF AUTOIMMUNE AND INFLAMMATORY DISEASES AEGERA THERAPEUTICS INC. (CA) 2011-03-31 WO disclosed