SCHEMBL12830278

SCHEMBL12830278

Nc1cccc(C(=O)Nc2cc(F)cc(Oc3cccnc3)c2)c1

nearest known ligand 0.68

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 5/20 0.58
SMN1; SMN2 Q16637 2/20 0.53
LMNA P02545 1/20 0.53
FFAR4 Q5NUL3 1/20 0.52
TSHR P16473 1/20 0.50
ALDH1A1 P00352 1/20 0.50
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
KMT2A Q03164 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12830298 0.89 GRM5 (0.56) GRM5
SCHEMBL4475675 0.89 TSHR (0.59) GRM5SMN1; SMN2LMNAFFAR4TSHR
SCHEMBL4478047 0.88 GRM5 (0.59) GRM5SMN1; SMN2LMNAFFAR4TSHR
SCHEMBL12830517 0.88 GRM5 (0.64) GRM5SMN1; SMN2LMNATSHRALDH1A1
SCHEMBL12830291 0.87 GRM5 (0.67) GRM5SMN1; SMN2LMNATSHRKMT2A
SCHEMBL12412147 0.87 GRM5 (0.61) GRM5SMN1; SMN2LMNATSHRALDH1A1
SCHEMBL12412646 0.87 GRM5 (0.77) GRM5KMT2A
SCHEMBL6926437 0.87 GRM5 (0.76) GRM5SMN1; SMN2LMNATSHRALDH1A1
SCHEMBL12830285 0.87 NPC1 (0.56) GRM5SMN1; SMN2LMNATSHRKMT2A
SCHEMBL12412157 0.85 GRM5 (0.63) GRM5SMN1; SMN2LMNAFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035214-A1 SUBSTITUTED PHENYLAMINE CARBOXAMIDE ANALOGS AS MGLUR5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSITY (US) 2011-03-24 WO disclosed