SCHEMBL6926437

SCHEMBL6926437

Nc1cccc(C(=O)Nc2cncc(Oc3cccnc3)c2)c1

nearest known ligand 0.76

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 7/20 0.76
ALDH1A1 P00352 1/20 0.57
SMN1; SMN2 Q16637 2/20 0.56
LMNA P02545 1/20 0.56
TSHR P16473 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12830517 0.92 GRM5 (0.64) GRM5ALDH1A1SMN1; SMN2LMNATSHR
SCHEMBL6926476 0.88 GRM5 (0.74) GRM5
SCHEMBL12830291 0.87 GRM5 (0.67) GRM5SMN1; SMN2LMNATSHR
SCHEMBL12830278 0.87 GRM5 (0.58) GRM5ALDH1A1SMN1; SMN2LMNATSHR
SCHEMBL12416360 0.86 GRM5 (0.76) GRM5ALDH1A1SMN1; SMN2LMNATSHR
SCHEMBL1487647 0.86 GRM5 (1.00) GRM5ALDH1A1
SCHEMBL6925812 0.86 GRM5 (1.00) GRM5ALDH1A1SMN1; SMN2LMNA
SCHEMBL12830285 0.84 NPC1 (0.56) GRM5SMN1; SMN2LMNATSHR
SCHEMBL7078083 0.84 LMNA (0.69) ALDH1A1LMNATSHR
SCHEMBL6926454 0.83 GRM5 (1.00) GRM5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035174-A1 SUBSTITUTED HETEROARYLAMINE CARBOXAMIDE ANALOGS AS MGLUR5 NEGATIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING THE SAME VANDERBILT UNIVERSITY (US) 2011-03-24 WO disclosed