SCHEMBL12831726

SCHEMBL12831726

COc1nc2c(C(F)(F)F)cccc2n1C(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 8/20 0.38
NR1H3 Q13133 8/20 0.38
ATM Q13315 3/20 0.37
MAPT P10636 2/20 0.37
TSHR P16473 1/20 0.37
MAPK1 P28482 1/20 0.37
CASP1 P29466 1/20 0.37
CASP7 P55210 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
GRM2 Q14416 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
F2RL3 Q96RI0 1/20 0.34
PDE2A O00408 1/20 0.34
PDE10A Q9Y233 1/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
HTR3A P46098 1/20 0.34
HSD11B1 P28845 2/20 0.33
TP53 P04637 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12730123 0.79 P2RX7 (0.41) NR1H2NR1H3ATMMAPTTSHR
SCHEMBL12792071 0.71 KMT2A (0.55) ATMMAPTTSHRMAPK1CASP1
SCHEMBL24910306 0.68 NR1H2 (0.47) NR1H2NR1H3GRM2PDE10AHTR3A
SCHEMBL10239600 0.66 KMT2A (0.38) ATMMAPTTSHRMAPK1CASP1
SCHEMBL1271026 0.65 NR1H2 (0.56) NR1H2NR1H3MAPTTSHRMEN1
SCHEMBL1272181 0.65 NR1H2 (0.56) NR1H2NR1H3MAPK1
SCHEMBL26375284 0.65 CYP1A2 (0.47) NR1H2NR1H3GRM2LMNAPDE10A
SCHEMBL1272253 0.64 NR1H2 (0.49) NR1H2NR1H3PDE2APDE10AHTR3A
SCHEMBL1272812 0.64 NR1H2 (0.67) NR1H2NR1H3MEN1KMT2A
SCHEMBL1271040 0.64 NR1H2 (0.67) NR1H2NR1H3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011038293-A1 CYCLIC PEPTIDE INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2011-03-31 WO disclosed