SCHEMBL12835898

SCHEMBL12835898

COC(=O)c1ccc(C[C@@H]2CC[C@H]([C@H](O)c3cccnc3)N2C(=O)OC(C)(C)C)cc1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
ADRB3 P13945 11/20 0.38
SLC6A4 P31645 1/20 0.38
MAPT P10636 1/20 0.37
GPR119 Q8TDV5 2/20 0.37
ALDH1A1 P00352 1/20 0.36
NAMPT P43490 1/20 0.36
ADRB1 P08588 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9934066 0.91 ADRB3 (0.40) ADRB3SLC6A4GPR119NAMPTADRB1
SCHEMBL9934063 0.91 ADRB3 (0.40) ADRB3SLC6A4GPR119NAMPTADRB1
SCHEMBL12862418 0.89 GPR119 (0.39) ADRB3SLC6A4GPR119NAMPT
SCHEMBL12862385 0.89 GPR119 (0.39) ADRB3SLC6A4GPR119NAMPT
SCHEMBL17986569 0.89 GPR119 (0.39) ADRB3SLC6A4GPR119NAMPT
SCHEMBL9934730 0.88 MAPT (0.42) ADRB3SLC6A4MAPTALDH1A1ADRB1
SCHEMBL9934734 0.88 MAPT (0.42) ADRB3SLC6A4MAPTALDH1A1ADRB1
SCHEMBL16619092 0.87 HDAC1 (0.38) HDAC1HDAC6SLC6A4MAPTGPR119
SCHEMBL18210791 0.87 HDAC1 (0.38) HDAC1HDAC6SLC6A4MAPTGPR119
SCHEMBL17986557 0.87 HDAC1 (0.38) HDAC1HDAC6SLC6A4MAPTGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011025690-A1 NOVEL PYRROLIDINE DERIVED BETA 3 ADRENERGIC RECEPTOR AGONISTS MERCK SHARP & DOHME CORP. (US) 2011-03-03 WO disclosed