SCHEMBL12875809

SCHEMBL12875809

N#Cc1cnn2nncc2c1Cl

nearest known ligand 0.34

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CDK2 P24941 2/20 0.31
CSNK1A1 P48729 1/20 0.30
CLK4 Q9HAZ1 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
POLB P06746 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9923108 0.79 KMT2A (0.38) CDK2KDM4EALDH1A1POLBRXFP1
SCHEMBL9923104 0.79 CDK2 (0.31) CDK2
SCHEMBL9923307 0.75 CDK2 (0.34) CDK2CSNK1A1CLK4KDM4EALDH1A1
SCHEMBL9923423 0.70 MEN1 (0.36) CDK2KDM4EALDH1A1LMNAPOLB
SCHEMBL9920417 0.69
SCHEMBL9923278 0.68 CDK2 (0.41) CDK2CSNK1A1CLK4KDM4EALDH1A1
SCHEMBL9923348 0.68 CDK2 (0.38) CDK2CSNK1A1CLK4KDM4EALDH1A1
SCHEMBL1160390 0.68 CDK2 (0.49) CDK2KDM4EALDH1A1
SCHEMBL9923105 0.67 PKM (0.34) ALDH1A1
SCHEMBL12492445 0.65 CDK2 (0.35) CDK2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2013033093-A1 HETEROCYCLIC COMPOUNDS AS JANUS KINASE INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2013-03-07 WO disclosed
WO-2011014817-A1 PYRROLO [1, 2-B] PYRIDAZINE DERIVATIVES AS JANUS KINASE INHIBITORS BIOCRYST PHARMACEUTICALS, INC. (US) 2011-02-03 WO disclosed