SCHEMBL12876196

SCHEMBL12876196

Cc1cc(Br)cc(-c2nc(COC3CCCCO3)c(C)s2)c1

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KDM4C Q9H3R0 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.31
ICAM1 P05362 1/20 0.31
SELE P16581 1/20 0.31
ALDH1A1 P00352 1/20 0.30
PPARG P37231 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1197708 0.88 PPARG (0.34) KDM4CNPC1RAB9AL3MBTL1PPARG
SCHEMBL12876229 0.86 NPC1 (0.34) KDM4CNPC1RAB9AL3MBTL1ICAM1
SCHEMBL12876224 0.85 PPARG (0.32) KDM4CNPC1RAB9AL3MBTL1ICAM1
SCHEMBL15006436 0.81 NPC1 (0.31) NPC1RAB9APPARGPPARA
SCHEMBL1198072 0.77 PPARG (0.34) KDM4CNPC1RAB9AL3MBTL1ICAM1
SCHEMBL1199086 0.76 PPARG (0.36) KDM4CL3MBTL1ICAM1SELEPPARG
SCHEMBL4724279 0.75 CREBBP (0.40) KDM4CNPC1RAB9AL3MBTL1ICAM1
SCHEMBL12876153 0.73 FFAR1 (0.38) KDM4CNPC1RAB9AICAM1SELE
SCHEMBL12876144 0.73 RAB9A (0.38) KDM4CNPC1RAB9AICAM1SELE
SCHEMBL12876150 0.73 FFAR1 (0.36) KDM4CNPC1RAB9AL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8461348-B2 Heterocyclic derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2013-06-11 US disclosed
US-20110028493-A1 HETEROCYCLIC DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-02-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110028493-A1 HETEROCYCLIC DERIVATIVE AND USE THEREOF PDE3B, PDE5A, PDE2A KDM4C 2736/4885NPC1 3877/4885RAB9A 2507/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.