SCHEMBL12880575

SCHEMBL12880575

BrC(c1ccc(C(Br)c2cccc3ccccc23)cc1)c1cccc2ccccc12

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.79
CYP1A2 P05177 3/20 0.79
CYP2C9 P11712 1/20 0.79
CYP2C19 P33261 1/20 0.79
SLC6A4 P31645 1/20 0.46
CYP2A6 P11509 3/20 0.40
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
ADRA2A P08913 4/20 0.39
ADRA2B P18089 4/20 0.39
ADRA2C P18825 4/20 0.39
ADRA1A P35348 4/20 0.39
ADRA1D P25100 3/20 0.39
ADRA1B P35368 3/20 0.39
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
KEAP1 Q14145 1/20 0.38
ACP3 P15309 1/20 0.38
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1643410 0.94 ALDH1A1 (0.76) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL11444158 0.89 ALDH1A1 (1.00) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL28192 0.79 ALDH1A1 (0.74) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL18242412 0.77 ALDH1A1 (0.71) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL28461729 0.76 ALDH1A1 (0.68) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL2332847 0.76 ALDH1A1 (0.68) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL9669273 0.75 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL6008494 0.75 ALDH1A1 (0.67) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL12880576 0.74 ALDH1A1 (0.54) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4
SCHEMBL2494544 0.74 ALDH1A1 (0.65) ALDH1A1CYP1A2CYP2C9CYP2C19SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7884175-B2 polymerizing one or more monomers containing dihalogen containing substituted biaryls, via a base-induced dehydrohalogenation MERCK PATENT GMBH (DE) 2011-02-08 US disclosed
US-7884175-B2 polymerizing one or more monomers containing dihalogen containing substituted biaryls, via a base-induced dehydrohalogenation MERCK PATENT GMBH (DE) 2011-02-08 US disclosed
EP-1623471-B1 METHOD FOR CONTROLLING THE MOLECULAR WEIGHT DURING POLY(ARYLENE VINYLENE) SYNTHESIS, AND POLYMERS PRODUCED THEREWITH MERCK PATENT GMBH (DE) 2007-05-30 EP disclosed