SCHEMBL129153

SCHEMBL129153

O=S(=O)(Oc1cccc(-c2cc3ccccc3cn2)c1)C(F)(F)F

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.44
RAB9A P51151 2/20 0.44
SDHB P21912 1/20 0.44
IDO1 P14902 1/20 0.43
TDO2 P48775 1/20 0.43
ADORA2A P29274 1/20 0.42
ADORA1 P30542 1/20 0.42
PDE4A P27815 3/20 0.41
PDE4C Q08493 3/20 0.41
PDE4D Q08499 3/20 0.41
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.40
PTGS1 P23219 1/20 0.39
PTGS2 P35354 1/20 0.39
ATR Q13535 1/20 0.38
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3810758 0.82 NPC1 (0.41) NPC1RAB9ASDHBADORA2AADORA1
SCHEMBL649550 0.81 GRM5 (0.46) NPC1RAB9ASDHBADORA2AADORA1
SCHEMBL4684800 0.79 PTPN1 (0.47) SDHBADORA2AADORA1CA1CA2
SCHEMBL13416088 0.79 CA1 (0.45) SDHBADORA2AADORA1PDE4APDE4C
SCHEMBL23956362 0.79 DYRK1A (0.40) SDHBADORA2AADORA1KDM4EALDH1A1
SCHEMBL649934 0.78 GRM5 (0.44) NPC1RAB9ASDHBADORA2AADORA1
SCHEMBL7608891 0.78 NPC1 (0.54) NPC1RAB9AIDO1TDO2KDM4E
SCHEMBL12072784 0.77 NPC1 (0.47) NPC1RAB9AIDO1TDO2
SCHEMBL127875 0.77 PDE4A (0.46) NPC1RAB9AADORA2AADORA1PDE4A
SCHEMBL18389050 0.76 ADORA2A (0.44) SDHBADORA2AADORA1PDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed
WO-2010127307-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2010-11-04 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120059026-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L NPC1 866/4885RAB9A 1144/4885SDHB 4162/4885
US-20140315939-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L NPC1 799/4885RAB9A 964/4885SDHB 4347/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.