SCHEMBL1291817

SCHEMBL1291817

COc1cc2[nH]c(=O)c(=O)[nH]c2cc1Cl

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN2D O15399 12/20 0.73
GRIN3B O60391 12/20 0.73
GRIN1 Q05586 12/20 0.73
GRIN2A Q12879 12/20 0.73
GRIN2B Q13224 12/20 0.73
GRIN2C Q14957 12/20 0.73
GRIN3A Q8TCU5 12/20 0.73
ALDH1A1 P00352 3/20 0.61
MAPT P10636 3/20 0.61
KDM4E B2RXH2 2/20 0.61
HPGD P15428 2/20 0.61
SMN1; SMN2 Q16637 2/20 0.61
GRIA1 P42261 2/20 0.61
LMNA P02545 2/20 0.61
MEN1 O00255 1/20 0.61
CYP1A2 P05177 1/20 0.61
TSHR P16473 1/20 0.61
THPO P40225 1/20 0.61
GRIA2 P42262 1/20 0.61
GRIA3 P42263 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1292034 0.85 GRIN2D (1.00) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL21360424 0.79 GRIN2D (0.50) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
2,3-Dihydroxy-6,7-Dichloroquinoxaline SCHEMBL30561497 0.78 GRIN2D (1.00) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
2,3-Dihydroxy-6,7-Dichloroquinoxaline SCHEMBL463608 0.78 GRIN2D (1.00) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL14326945 0.78 GRIN2D (0.76) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL10955203 0.77 ALDH1A1 (0.75) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL22186137 0.77 IDH1 (0.57) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL18308359 0.76 GRIN2D (0.73) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL21676446 0.76 GRIN2D (0.73) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL5155436 0.76 GRIN2D (0.73) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012045196-A1 PHOSPHOGLYCERATE KINASE INHIBITORS ABBOTT LABORATORIES (US) 2012-04-12 WO disclosed