SCHEMBL12933335

SCHEMBL12933335

CCn1c(=O)n(CC(C)(C)C)c(=O)c2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PGR P06401 2/20 0.57
MAPK8 P45983 1/20 0.54
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 5/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
KMT2A Q03164 2/20 0.50
RCE1 Q9Y256 1/20 0.50
RECQL P46063 1/20 0.50
CNR2 P34972 3/20 0.49
TP53 P04637 1/20 0.49
HSD17B10 Q99714 1/20 0.46
MAPK1 P28482 1/20 0.46
MDM2 Q00987 1/20 0.46
HDAC1 Q13547 1/20 0.46
RORA P35398 1/20 0.45
RORC P51449 1/20 0.45
RORB Q92753 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30485670 0.87 PGR (0.68) PGRMAPK8ALDH1A1KDM4ESMN1; SMN2
SCHEMBL6362477 0.87 PGR (0.68) PGRMAPK8ALDH1A1KDM4ESMN1; SMN2
SCHEMBL12933336 0.81 TOP2A (0.51) PGRALDH1A1KDM4ECNR2HDAC1
SCHEMBL12963428 0.81 PGR (0.61) PGRMAPK8ALDH1A1KDM4ESMN1; SMN2
SCHEMBL12933344 0.81 PARG (0.43) PGRALDH1A1KDM4ESMN1; SMN2KMT2A
SCHEMBL12933334 0.77 GAA (0.52) ALDH1A1SMN1; SMN2KMT2ACNR2HDAC1
SCHEMBL12933342 0.77 P2RX4 (0.62) SMN1; SMN2KMT2ATP53MAPK1HDAC1
SCHEMBL6366020 0.77 PGR (0.64) PGRMAPK8ALDH1A1KDM4ESMN1; SMN2
SCHEMBL16092741 0.76 PGR (0.55) PGRMAPK8ALDH1A1KDM4ESMN1; SMN2
SCHEMBL13111957 0.75 CYP1A2 (0.56) ALDH1A1KDM4EKMT2AHSD17B10MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7868204-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2011-01-11 US disclosed
US-7838520-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2010-11-23 US disclosed
US-7595343-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2009-09-29 US disclosed
US-7595343-B2 Inhibitors of histone deacetylase METHYLGENE, INC. (CA) 2009-09-29 US disclosed